Abstract
The synthesis of 6β-(methylfumaramido) and 6β-chloroacetamido derivatives 1b and 1c of 6β-amino-7,8-didehydromorphinan and the corresponding 14-hydroxy derivatives 1e and 1f are described. The 7,8-dihydro derivatives of these compounds were synthesized in inactive (2b, c, e, f) as well as in tritiated form (3b, c, e, f).
| Original language | English |
|---|---|
| Pages (from-to) | 133-136 |
| Number of pages | 4 |
| Journal | Helvetica Chimica Acta |
| Volume | 79 |
| Issue number | 1 |
| Publication status | Published - 1996 |
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All Science Journal Classification (ASJC) codes
- Chemistry(all)
Cite this
Ötvös, F., Tóth, G., Lovas, S., Simon, C., & Hosztafi, S. (1996). 13. Synthesis and tritium labelling of 6β-amino-4,5α-epoxyraorphinans and their 14-hydroxy derivatives as potential affinity labelling probes with μ opioid agonist activity. Helvetica Chimica Acta, 79(1), 133-136.