Abstract
The synthesis of 6β-(methylfumaramido) and 6β-chloroacetamido derivatives 1b and 1c of 6β-amino-7,8-didehydromorphinan and the corresponding 14-hydroxy derivatives 1e and 1f are described. The 7,8-dihydro derivatives of these compounds were synthesized in inactive (2b, c, e, f) as well as in tritiated form (3b, c, e, f).
| Original language | English (US) |
|---|---|
| Pages (from-to) | 133-136 |
| Number of pages | 4 |
| Journal | Helvetica Chimica Acta |
| Volume | 79 |
| Issue number | 1 |
| DOIs | |
| State | Published - Jan 1 1996 |
All Science Journal Classification (ASJC) codes
- Catalysis
- Biochemistry
- Drug Discovery
- Physical and Theoretical Chemistry
- Organic Chemistry
- Inorganic Chemistry
Fingerprint Dive into the research topics of '13. Synthesis and tritium labelling of 6β-amino-4,5α-epoxyraorphinans and their 14-hydroxy derivatives as potential affinity labelling probes with μ opioid agonist activity'. Together they form a unique fingerprint.
Cite this
Ötvös, F., Tóth, G., Lovas, S., Simon, C., & Hosztafi, S. (1996). 13. Synthesis and tritium labelling of 6β-amino-4,5α-epoxyraorphinans and their 14-hydroxy derivatives as potential affinity labelling probes with μ opioid agonist activity. Helvetica Chimica Acta, 79(1), 133-136. https://doi.org/10.1002/hlca.19960790114