Abstract
The synthesis of 6β-(methylfumaramido) and 6β-chloroacetamido derivatives 1b and 1c of 6β-amino-7,8-didehydromorphinan and the corresponding 14-hydroxy derivatives 1e and 1f are described. The 7,8-dihydro derivatives of these compounds were synthesized in inactive (2b, c, e, f) as well as in tritiated form (3b, c, e, f).
| Original language | English |
|---|---|
| Pages (from-to) | 133-136 |
| Number of pages | 4 |
| Journal | Helvetica Chimica Acta |
| Volume | 79 |
| Issue number | 1 |
| State | Published - 1996 |
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All Science Journal Classification (ASJC) codes
- Chemistry(all)
Cite this
13. Synthesis and tritium labelling of 6β-amino-4,5α-epoxyraorphinans and their 14-hydroxy derivatives as potential affinity labelling probes with μ opioid agonist activity. / Ötvös, Ferenc; Tóth, Géza; Lovas, Sándor; Simon, Csaba; Hosztafi, Sándor.
In: Helvetica Chimica Acta, Vol. 79, No. 1, 1996, p. 133-136.Research output: Contribution to journal › Article
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TY - JOUR
T1 - 13. Synthesis and tritium labelling of 6β-amino-4,5α-epoxyraorphinans and their 14-hydroxy derivatives as potential affinity labelling probes with μ opioid agonist activity
AU - Ötvös, Ferenc
AU - Tóth, Géza
AU - Lovas, Sándor
AU - Simon, Csaba
AU - Hosztafi, Sándor
PY - 1996
Y1 - 1996
N2 - The synthesis of 6β-(methylfumaramido) and 6β-chloroacetamido derivatives 1b and 1c of 6β-amino-7,8-didehydromorphinan and the corresponding 14-hydroxy derivatives 1e and 1f are described. The 7,8-dihydro derivatives of these compounds were synthesized in inactive (2b, c, e, f) as well as in tritiated form (3b, c, e, f).
AB - The synthesis of 6β-(methylfumaramido) and 6β-chloroacetamido derivatives 1b and 1c of 6β-amino-7,8-didehydromorphinan and the corresponding 14-hydroxy derivatives 1e and 1f are described. The 7,8-dihydro derivatives of these compounds were synthesized in inactive (2b, c, e, f) as well as in tritiated form (3b, c, e, f).
UR - http://www.scopus.com/inward/record.url?scp=0041022342&partnerID=8YFLogxK
UR - http://www.scopus.com/inward/citedby.url?scp=0041022342&partnerID=8YFLogxK
M3 - Article
AN - SCOPUS:0041022342
VL - 79
SP - 133
EP - 136
JO - Helvetica Chimica Acta
JF - Helvetica Chimica Acta
SN - 0018-019X
IS - 1
ER -